BRL 44408 ( BRL44408;BRL-44408 )

Catalog No. M10622 CAS No. 118343-19-4

A potent, selective α2A-adrenoceptor antagonist with Ki of 1.7 nM, 80-fold selectivity over α2B-adrenergic receptors.

Purity : >98% (HPLC)

COA

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HPLC

MSDS

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Biological Information

Product Name

BRL 44408
Note

Research use only, not for human use.
Brief Description

A potent, selective α2A-adrenoceptor antagonist with Ki of 1.7 nM, 80-fold selectivity over α2B-adrenergic receptors.
Description

A potent, selective α2A-adrenoceptor antagonist with Ki of 1.7 nM, 80-fold selectivity over α2B-adrenergic receptors; significantly increases stimulated noradrenaline release in rat locus coeruleus slices at 0.1-1 uM, significantly increases the electrically induced release in rats.
Synonyms

BRL44408;BRL-44408
Pathway

Angiogenesis
Target

Adrenergic Receptor
Recptor

Adrenergic Receptor
Research Area

——
Indication

——

Chemical Information

CAS Number

118343-19-4
Formula Weight

215.30
Molecular Formula

C13H17N3
Purity

>98% (HPLC)
Solubility

——
SMILES

CC1C2=CC=CC=C2CN1CC3=NCCN3
Chemical Name

2-((4,5-dihydro-1H-imidazol-2-yl)methyl)-2,3-dihydro-1-methyl-1H-isoindole

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Kiss JP, et al. Brain Res. 1995 Mar 20;674(2):238-44.
2. Callado LF, et al. Eur J Pharmacol. 1999 Jan 29;366(1):35-9.
3. Young P, et al. Eur J Pharmacol. 1989 Sep 22;168(3):381-6.

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